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TargetSignal transducer and activator of transcription 3 [702-738,740-752]
LigandBDBM46350
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based assay to measure STAT3 inhibition
IC50 2901±n/a nM
Citation PubChem, PC Dose response cell-based assay to measure STAT3 inhibition PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Signal transducer and activator of transcription 3 [702-738,740-752]
Name:Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:APRF | STAT3 | STAT3_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:5263.93
Organism:Homo sapiens (Human)
Description:gi_13272532
Residue:50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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BDBM46350
n/a
NameBDBM46350
Synonyms:4-[[4-(morpholinomethyl)benzoyl]amino]benzoic acid ethyl ester | 4-[[[4-(4-morpholinylmethyl)phenyl]-oxomethyl]amino]benzoic acid ethyl ester | MLS000061256 | SMR000070125 | cid_1257531 | ethyl 4-[[4-(morpholin-4-ylmethyl)benzoyl]amino]benzoate | ethyl 4-[[4-(morpholin-4-ylmethyl)phenyl]carbonylamino]benzoate | ethyl 4-{[4-(4-morpholinylmethyl)benzoyl]amino}benzoate
TypeSmall organic molecule
Emp. Form.C21H24N2O4
Mol. Mass.368.4263
SMILESCCOC(=O)c1ccc(NC(=O)c2ccc(CN3CCOCC3)cc2)cc1
Structure
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