| Reaction Details |
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 | Report a problem with these data |
| Target | Signal transducer and activator of transcription 3 [702-738,740-752] |
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| Ligand | BDBM43521 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response counterscreen for STAT1 inhibitors: cell-based high throughput assay to measure STAT3 inhibition |
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| IC50 | >55700±n/a nM |
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| Citation |  PubChem, PC Dose response counterscreen for STAT1 inhibitors: cell-based high throughput assay to measure STAT3 inhibition PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Signal transducer and activator of transcription 3 [702-738,740-752] |
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| Name: | Signal transducer and activator of transcription 3 [702-738,740-752] |
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| Synonyms: | APRF | STAT3 | STAT3_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 5263.93 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_13272532 |
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| Residue: | 50 |
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| Sequence: | AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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| BDBM43521 |
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| n/a |
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| Name | BDBM43521 |
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| Synonyms: | MLS000394345 | N-(4-fluorophenyl)-2-[4-(4-methylphenyl)sulfonyl-1-piperazinyl]-2-phenylacetamide | N-(4-fluorophenyl)-2-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]-2-phenyl-ethanamide | N-(4-fluorophenyl)-2-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]-2-phenylacetamide | N-(4-fluorophenyl)-2-phenyl-2-(4-tosylpiperazino)acetamide | SMR000248320 | cid_15945370 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H26FN3O3S |
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| Mol. Mass. | 467.556 |
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| SMILES | Cc1ccc(cc1)S(=O)(=O)N1CCN(CC1)C(C(=O)Nc1ccc(F)cc1)c1ccccc1 |
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| Structure | 
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