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TargetMucolipin-3
LigandBDBM46854
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based high-throughput screening assay for agonists of the transient receptor potential channel ML3 (TRPML3)
EC50 3580±n/a nM
Citation PubChem, PC Dose response cell-based high-throughput screening assay for agonists of the transient receptor potential channel ML3 (TRPML3) PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Mucolipin-3
Name:Mucolipin-3
Synonyms:MCLN3_HUMAN | MCOLN3 | MCOLN3 protein
Type:Enzyme Catalytic Domain
Mol. Mass.:64244.09
Organism:Homo sapiens (Human)
Description:Q8TDD5
Residue:553
Sequence:
MADPEVVVSSCSSHEEENRCNFNQQTSPSEELLLEDQMRRKLKFFFMNPCEKFWARGRKP
WKLAIQILKIAMVTIQLVLFGLSNQMVVAFKEENTIAFKHLFLKGYMDRMDDTYAVYTQS
DVYDQLIFAVNQYLQLYNVSVGNHAYENKGTKQSAMAICQHFYKRGNIYPGNDTFDIDPE
IETECFFVEPDEPFHIGTPAENKLNLTLDFHRLLTVELQFKLKAINLQTVRHQELPDCYD
FTLTITFDNKAHSGRIKISLDNDISIRECKDWHVSGSIQKNTHYMMIFDAFVILTCLVSL
ILCIRSVIRGLQLQQEFVNFFLLHYKKEVSVSDQMEFVNGWYIMIIISDILTIIGSILKM
EIQAKSLTSYDVCSILLGTSTMLVWLGVIRYLGFFAKYNLLILTLQAALPNVIRFCCCAA
MIYLGYCFCGWIVLGPYHDKFRSLNMVSECLFSLINGDDMFATFAKMQQKSYLVWLFSRI
YLYSFISLFIYMILSLFIALITDTYETIKQYQQDGFPETELRTFISECKDLPNSGKYRLE
DDPPVSLFCCCKK
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  Blast E-value cutoff:
BDBM46854
n/a
NameBDBM46854
Synonyms:1-(2,5-dimethoxyphenyl)sulfonyl-3,4-dihydro-2H-quinoline | MLS000113521 | SMR000109419 | cid_778296
TypeSmall organic molecule
Emp. Form.C17H19NO4S
Mol. Mass.333.402
SMILESCOc1ccc(OC)c(c1)S(=O)(=O)N1CCCc2ccccc12
Structure
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