| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Regulator of G-protein signaling 8 |
|---|
| Ligand | BDBM47778 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao. |
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| EC50 | >30000±n/a nM |
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| Citation |  PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Regulator of G-protein signaling 8 |
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| Name: | Regulator of G-protein signaling 8 |
|---|
| Synonyms: | RGS8 | RGS8_HUMAN | Regulator of G-protein signaling 8 (RGS8) |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 20925.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_74355113 |
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| Residue: | 180 |
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| Sequence: | MAALLMPRRNKGMRTRLGCLSHKSDSCSDFTAILPDKPNRALKRLSTEEATRWADSFDVL
LSHKYGVAAFRAFLKTEFSEENLEFWLACEEFKKTRSTAKLVSKAHRIFEEFVDVQAPRE
VNIDFQTREATRKNLQEPSLTCFDQAQGKVHSLMEKDSYPRFLRSKMYLDLLSQSQRRLS
|
|
|
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| BDBM47778 |
|---|
| n/a |
|---|
| Name | BDBM47778 |
|---|
| Synonyms: | 1-(2-methoxy-5-methyl-phenyl)-3-(3-methoxyphenyl)urea | 1-(2-methoxy-5-methylphenyl)-3-(3-methoxyphenyl)urea | MLS000679289 | N-(2-methoxy-5-methylphenyl)-N'-(3-methoxyphenyl)urea | SMR000297699 | cid_6467994 |
|---|
| Type | Small organic molecule |
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| Emp. Form. | C16H18N2O3 |
|---|
| Mol. Mass. | 286.3257 |
|---|
| SMILES | COc1cccc(NC(=O)Nc2cc(C)ccc2OC)c1 |
|---|
| Structure | 
|
|---|
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