| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Regulator of G-protein signaling 8 |
|---|
| Ligand | BDBM47816 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao. |
|---|
| EC50 | 4250±n/a nM |
|---|
| Citation |  PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao. PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Regulator of G-protein signaling 8 |
|---|
| Name: | Regulator of G-protein signaling 8 |
|---|
| Synonyms: | RGS8 | RGS8_HUMAN | Regulator of G-protein signaling 8 (RGS8) |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 20925.80 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_74355113 |
|---|
| Residue: | 180 |
|---|
| Sequence: | MAALLMPRRNKGMRTRLGCLSHKSDSCSDFTAILPDKPNRALKRLSTEEATRWADSFDVL
LSHKYGVAAFRAFLKTEFSEENLEFWLACEEFKKTRSTAKLVSKAHRIFEEFVDVQAPRE
VNIDFQTREATRKNLQEPSLTCFDQAQGKVHSLMEKDSYPRFLRSKMYLDLLSQSQRRLS
|
|
|
|---|
| BDBM47816 |
|---|
| n/a |
|---|
| Name | BDBM47816 |
|---|
| Synonyms: | 6-Oxo-6H-anthra[1,9-cd]isoxazole-3-carboxylic acid (3-methoxy-propyl)-amide | MLS001029502 | SMR000425486 | cid_3729555 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H16N2O4 |
|---|
| Mol. Mass. | 336.3413 |
|---|
| SMILES | COCCCNC(=O)c1ccc2C(=O)c3ccccc3-c3onc1c23 |
|---|
| Structure | 
|
|---|
Search and Browse
