| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 7 |
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| Ligand | BDBM47724 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS7-Galphao. |
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| EC50 | >30000±n/a nM |
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| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS7-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Regulator of G-protein signaling 7 |
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| Name: | Regulator of G-protein signaling 7 |
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| Synonyms: | RGS7 | RGS7_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 57675.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49802 |
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| Residue: | 495 |
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| Sequence: | MAQGNNYGQTSNGVADESPNMLVYRKMEDVIARMQDEKNGIPIRTVKSFLSKIPSVFSGS
DIVQWLIKNLTIEDPVEALHLGTLMAAHGYFFPISDHVLTLKDDGTFYRFQTPYFWPSNC
WEPENTDYAVYLCKRTMQNKARLELADYEAESLARLQRAFARKWEFIFMQAEAQAKVDKK
RDKIERKILDSQERAFWDVHRPVPGCVNTTEVDIKKSSRMRNPHKTRKSVYGLQNDIRSH
SPTHTPTPETKPPTEDELQQQIKYWQIQLDRHRLKMSKVADSLLSYTEQYLEYDPFLLPP
DPSNPWLSDDTTFWELEASKEPSQQRVKRWGFGMDEALKDPVGREQFLKFLESEFSSENL
RFWLAVEDLKKRPIKEVPSRVQEIWQEFLAPGAPSAINLDSKSYDKTTQNVKEPGRYTFE
DAQEHIYKLMKSDSYPRFIRSSAYQELLQAKKKSGNSMDRRTSFEKFAQNVGRNIPIFPC
HKNCTPTLRASTNLL
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| BDBM47724 |
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| n/a |
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| Name | BDBM47724 |
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| Synonyms: | MLS000569357 | SMR000154979 | [1-[4-[(2-bromobenzoyl)amino]phenyl]imidazol-2-yl]-phenyl-phosphinic acid | [1-[4-[(2-bromobenzoyl)amino]phenyl]imidazol-2-yl]-phenylphosphinic acid | [1-[4-[(2-bromophenyl)carbonylamino]phenyl]imidazol-2-yl]-phenyl-phosphinic acid | [1-[4-[[(2-bromophenyl)-oxomethyl]amino]phenyl]-2-imidazolyl]-phenylphosphinic acid | cid_5207778 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H17BrN3O3P |
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| Mol. Mass. | 482.266 |
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| SMILES | OP(=O)(c1nccn1-c1ccc(NC(=O)c2ccccc2Br)cc1)c1ccccc1 |
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| Structure | 
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