| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 19 |
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| Ligand | BDBM41758 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. |
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| EC50 | >30000±n/a nM |
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| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Regulator of G-protein signaling 19 |
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| Name: | Regulator of G-protein signaling 19 |
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| Synonyms: | G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19) |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 24631.38 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_86990435 |
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| Residue: | 217 |
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| Sequence: | MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQ
ASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFW
LACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDA
QLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
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| BDBM41758 |
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| n/a |
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| Name | BDBM41758 |
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| Synonyms: | (2-{2-[5-(4-Fluoro-phenyl)-[1,3,4]oxadiazol-2-ylsulfanyl]-acetylamino}-thiazol-4-yl)-acetic acid ethyl ester | 2-[2-[[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl ester | 2-[2-[[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]thio]acetyl]amino]thiazol-4-yl]acetic acid ethyl ester | MLS000071801 | SMR000003120 | cid_653271 | ethyl 2-[2-[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethanoylamino]-1,3-thiazol-4-yl]ethanoate | ethyl 2-[2-[[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]amino]-1,3-thiazol-4-yl]acetate |
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| Type | Small organic molecule |
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| Emp. Form. | C17H15FN4O4S2 |
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| Mol. Mass. | 422.454 |
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| SMILES | CCOC(=O)Cc1csc(NC(=O)CSc2nnc(o2)-c2ccc(F)cc2)n1 |
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| Structure | 
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