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TargetRegulator of G-protein signaling 19
LigandBDBM47708
Substrate/Competitorn/a
Meas. Tech.Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao.
EC50>30000±n/a nM
Citation PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Regulator of G-protein signaling 19
Name:Regulator of G-protein signaling 19
Synonyms:G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19)
Type:Enzyme Catalytic Domain
Mol. Mass.:24631.38
Organism:Homo sapiens (Human)
Description:gi_86990435
Residue:217
Sequence:
MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQ
ASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFW
LACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDA
QLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
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  Blast E-value cutoff:
BDBM47708
n/a
NameBDBM47708
Synonyms:1-(4-chlorobenzyl)sulfonylisonipecotic acid ethyl ester | 1-[(4-chlorophenyl)methylsulfonyl]-4-piperidinecarboxylic acid ethyl ester | MLS000066348 | SMR000081233 | cid_2228514 | ethyl 1-[(4-chlorobenzyl)sulfonyl]-4-piperidinecarboxylate | ethyl 1-[(4-chlorophenyl)methylsulfonyl]piperidine-4-carboxylate
TypeSmall organic molecule
Emp. Form.C15H20ClNO4S
Mol. Mass.345.842
SMILESCCOC(=O)C1CCN(CC1)S(=O)(=O)Cc1ccc(Cl)cc1
Structure
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