BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetRegulator of G-protein signaling 19
LigandBDBM47717
Substrate/Competitorn/a
Meas. Tech.Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao.
EC50>30000±n/a nM
Citation PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Regulator of G-protein signaling 19
Name:Regulator of G-protein signaling 19
Synonyms:G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19)
Type:Enzyme Catalytic Domain
Mol. Mass.:24631.38
Organism:Homo sapiens (Human)
Description:gi_86990435
Residue:217
Sequence:
MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQ
ASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFW
LACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDA
QLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM47717
n/a
NameBDBM47717
Synonyms:5-Ethylamino-anthra[1,9-cd]isoxazol-6-one | MLS000525596 | SMR000116070 | cid_776361
TypeSmall organic molecule
Emp. Form.C16H12N2O2
Mol. Mass.264.2787
SMILESCCNc1ccc2noc3-c4ccccc4C(=O)c1c23
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: