Reaction Details |
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Target | Regulator of G-protein signaling 19 |
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Ligand | BDBM46608 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. |
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EC50 | 1690±n/a nM |
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Citation | PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay(2009)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Regulator of G-protein signaling 19 |
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Name: | Regulator of G-protein signaling 19 |
Synonyms: | G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19) |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 24631.38 |
Organism: | Homo sapiens (Human) |
Description: | gi_86990435 |
Residue: | 217 |
Sequence: | MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQ
ASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFW
LACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDA
QLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
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BDBM46608 |
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n/a |
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Name | BDBM46608 |
Synonyms: | (4E)-5-methyl-4-[(3-nitroanilino)methylene]-2-phenyl-2-pyrazoline-3-thione | (4E)-5-methyl-4-[(3-nitroanilino)methylidene]-2-phenyl-3-pyrazolethione | (4E)-5-methyl-4-[(3-nitroanilino)methylidene]-2-phenylpyrazole-3-thione | (4E)-5-methyl-4-[[(3-nitrophenyl)amino]methylidene]-2-phenyl-pyrazole-3-thione | (4Z)-5-methyl-4-[(3-nitroanilino)methylene]-2-phenyl-2-pyrazoline-3-thione | MLS-0100444.0001 | cid_6945186 |
Type | Small organic molecule |
Emp. Form. | C17H14N4O2S |
Mol. Mass. | 338.384 |
SMILES | Cc1[n-]n(-c2ccccc2)c(=S)c1\C=[NH+]\c1cccc(c1)[N+]([O-])=O |
Structure |
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