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TargetRegulator of G-protein signaling 16
LigandBDBM47700
Substrate/Competitorn/a
Meas. Tech.Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao.
EC50>30000±n/a nM
Citation PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Regulator of G-protein signaling 16
Name:Regulator of G-protein signaling 16
Synonyms:RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16
Type:Enzyme Catalytic Domain
Mol. Mass.:22748.87
Organism:Homo sapiens (Human)
Description:gi_156416009
Residue:202
Sequence:
MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVL
GWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEE
FICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDL
AAQASAASATLSSCSLDEPSHT
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  Blast E-value cutoff:
BDBM47700
n/a
NameBDBM47700
Synonyms:2-(4-methyl-1-piperidinyl)aniline | 2-(4-methylpiperidin-1-yl)aniline | MLS000080408 | SMR000035930 | [2-(4-methylpiperidino)phenyl]amine | cid_663698
TypeSmall organic molecule
Emp. Form.C12H18N2
Mol. Mass.190.2847
SMILESCC1CCN(CC1)c1ccccc1N
Structure
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