| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 16 |
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| Ligand | BDBM47713 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. |
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| EC50 | >30000±n/a nM |
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| Citation |  PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Regulator of G-protein signaling 16 |
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| Name: | Regulator of G-protein signaling 16 |
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| Synonyms: | RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 22748.87 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_156416009 |
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| Residue: | 202 |
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| Sequence: | MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVL
GWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEE
FICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDL
AAQASAASATLSSCSLDEPSHT
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| BDBM47713 |
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| n/a |
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| Name | BDBM47713 |
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| Synonyms: | MLS000113446 | N-(1,5-dimethyl-3-oxidanylidene-2-phenyl-pyrazol-4-yl)-3,4-dimethoxy-N-methyl-benzenesulfonamide | N-(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)-3,4-dimethoxy-N-methylbenzenesulfonamide | N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3,4-dimethoxy-N-methylbenzenesulfonamide | N-(3-keto-1,5-dimethyl-2-phenyl-3-pyrazolin-4-yl)-3,4-dimethoxy-N-methyl-benzenesulfonamide | SMR000109344 | cid_1075678 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H23N3O5S |
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| Mol. Mass. | 417.479 |
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| SMILES | COc1ccc(cc1OC)S(=O)(=O)N(C)c1c(C)n(C)n(-c2ccccc2)c1=O |
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| Structure | 
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