| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 16 |
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| Ligand | BDBM47779 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. |
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| EC50 | >30000±n/a nM |
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| Citation |  PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Regulator of G-protein signaling 16 |
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| Name: | Regulator of G-protein signaling 16 |
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| Synonyms: | RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 22748.87 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_156416009 |
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| Residue: | 202 |
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| Sequence: | MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVL
GWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEE
FICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDL
AAQASAASATLSSCSLDEPSHT
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| BDBM47779 |
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| n/a |
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| Name | BDBM47779 |
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| Synonyms: | 2-furanyl-[4-[3-(4-morpholinyl)-4-nitrophenyl]-1-piperazinyl]methanone | 2-furyl-[4-(3-morpholino-4-nitro-phenyl)piperazino]methanone | MLS000711509 | SMR000281276 | cid_2894898 | furan-2-yl-[4-(3-morpholin-4-yl-4-nitro-phenyl)piperazin-1-yl]methanone | furan-2-yl-[4-(3-morpholin-4-yl-4-nitrophenyl)piperazin-1-yl]methanone |
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| Type | Small organic molecule |
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| Emp. Form. | C19H22N4O5 |
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| Mol. Mass. | 386.4018 |
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| SMILES | [O-][N+](=O)c1ccc(cc1N1CCOCC1)N1CCN(CC1)C(=O)c1ccco1 |
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| Structure | 
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