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TargetDual specificity protein phosphatase 3
LigandBDBM46208
Substrate/Competitorn/a
Meas. Tech.SAR VHR1 Fluorescent Assay for In Vitro dose response studies
IC50>99000±n/a nM
Citation PubChem, PC SAR VHR1 Fluorescent Assay for In Vitro dose response studies PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Dual specificity protein phosphatase 3
Name:Dual specificity protein phosphatase 3
Synonyms:DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR
Type:Hydrolase
Mol. Mass.:20480.58
Organism:Homo sapiens (Human)
Description:n/a
Residue:185
Sequence:
MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
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  Blast E-value cutoff:
BDBM46208
n/a
NameBDBM46208
Synonyms:(4-amino-3-p-phenetyl-2-thioxo-4-thiazolin-5-yl)-(4-methylpiperazino)methanone | MLS-0267194.0001 | [4-amino-3-(4-ethoxyphenyl)-2-sulfanylidene-1,3-thiazol-5-yl]-(4-methylpiperazin-1-yl)methanone | [4-amino-3-(4-ethoxyphenyl)-2-sulfanylidene-5-thiazolyl]-(4-methyl-1-piperazinyl)methanone | [4-azanyl-3-(4-ethoxyphenyl)-2-sulfanylidene-1,3-thiazol-5-yl]-(4-methylpiperazin-1-yl)methanone | cid_1545986
TypeSmall organic molecule
Emp. Form.C17H22N4O2S2
Mol. Mass.378.512
SMILESCCOc1ccc(cc1)-n1c(N)c(sc1=S)C(=O)N1CCN(C)CC1
Structure
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