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TargetDual specificity protein phosphatase 3
LigandBDBM46250
Substrate/Competitorn/a
Meas. Tech.SAR VHR1 Fluorescent Assay for In Vitro dose response studies
IC50 18300±n/a nM
Citation PubChem, PC SAR VHR1 Fluorescent Assay for In Vitro dose response studies PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Dual specificity protein phosphatase 3
Name:Dual specificity protein phosphatase 3
Synonyms:DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR
Type:Hydrolase
Mol. Mass.:20480.58
Organism:Homo sapiens (Human)
Description:n/a
Residue:185
Sequence:
MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
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BDBM46250
n/a
NameBDBM46250
Synonyms:(4E)-2-methoxy-4-[(pentan-3-ylamino)-sulfanyl-methylidene]cyclohexa-2,5-dien-1-one | (4E)-2-methoxy-4-[(pentan-3-ylamino)-sulfanylmethylidene]cyclohexa-2,5-dien-1-one | (4E)-4-[(1-ethylpropylamino)-mercapto-methylene]-2-methoxy-cyclohexa-2,5-dien-1-one | (4E)-4-[mercapto-(pentan-3-ylamino)methylidene]-2-methoxy-1-cyclohexa-2,5-dienone | MLS-0412118.0001 | cid_44182131
TypeSmall organic molecule
Emp. Form.C13H19NO2S
Mol. Mass.253.36
SMILESCCC(CC)NC(=S)c1ccc(O)c(OC)c1
Structure
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