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TargetDual specificity protein phosphatase 3
LigandBDBM46204
Substrate/Competitorn/a
Meas. Tech.SAR VHR1 absorbance Assay for In Vitro dose response studies.
IC50>100000±n/a nM
Citation PubChem, PC SAR VHR1 absorbance Assay for In Vitro dose response studies. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Dual specificity protein phosphatase 3
Name:Dual specificity protein phosphatase 3
Synonyms:DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR
Type:Hydrolase
Mol. Mass.:20480.58
Organism:Homo sapiens (Human)
Description:n/a
Residue:185
Sequence:
MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
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BDBM46204
n/a
NameBDBM46204
Synonyms:(4Z)-2-methoxy-4-[(4-methylpiperidin-1-yl)-sulfanyl-methylidene]cyclohexa-2,5-dien-1-one | (4Z)-2-methoxy-4-[(4-methylpiperidin-1-yl)-sulfanylmethylidene]cyclohexa-2,5-dien-1-one | (4Z)-4-[mercapto-(4-methyl-1-piperidinyl)methylidene]-2-methoxy-1-cyclohexa-2,5-dienone | (4Z)-4-[mercapto-(4-methylpiperidino)methylene]-2-methoxy-cyclohexa-2,5-dien-1-one | MLS-0078446.0001 | cid_5347726
TypeSmall organic molecule
Emp. Form.C14H19NO2S
Mol. Mass.265.371
SMILESCOc1cc(ccc1O)C(=S)N1CCC(C)CC1
Structure
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