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TargetTranscription factor p65
LigandBDBM49596
Substrate/Competitorn/a
Meas. Tech.Name: High Throughput Screen to Identify Compounds that increase expression of NF-kB in Human Neuronal Cells - Dose Response
EC50 319±n/a nM
Citation PubChem, PC Name: High Throughput Screen to Identify Compounds that increase expression of NF-kB in Human Neuronal Cells - Dose Response PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Transcription factor p65
Name:Transcription factor p65
Synonyms:NFKB3 | Nuclear factor NF-kappa-B | Nuclear factor NF-kappa-B p65 subunit | RELA | TF65_HUMAN | v-rel reticuloendotheliosis viral oncogene homolog A isoform 1
Type:Enzyme
Mol. Mass.:60211.92
Organism:Homo sapiens (Human)
Description:Q04206
Residue:551
Sequence:
MDELFPLIFPAEPAQASGPYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPT
IKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGFYEAELCPDRCIHSFQNLGIQC
VKKRDLEQAISQRIQTNNNPFQVPIEEQRGDYDLNAVRLCFQVTVRDPSGRPLRLPPVLS
HPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFS
QADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPDTDDRHRIEE
KRKRTYETFKSIMKKSPFSGPTDPRPPPRRIAVPSRSSASVPKPAPQPYPFTSSLSTINY
DEFPTMVFPSGQISQASALAPAPPQVLPQAPAPAPAPAMVSALAQAPAPVPVLAPGPPQA
VAPPAPKPTQAGEGTLSEALLQLQFDDEDLGALLGNSTDPAVFTDLASVDNSEFQQLLNQ
GIPVAPHTTEPMLMEYPEAITRLVTGAQRPPDPAPAPLGAPGLPNGLLSGDEDFSSIADM
DFSALLSQISS
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM49596
n/a
NameBDBM49596
Synonyms:2-[(E)-2-(2-fluorophenyl)ethenyl]quinoline | 2-[(E)-2-(2-fluorophenyl)vinyl]quinoline | 2-[2-(2-Fluoro-phenyl)-vinyl]-quinoline | MLS000561645 | SMR000176854 | cid_5763302
TypeSmall organic molecule
Emp. Form.C17H12FN
Mol. Mass.249.2823
SMILESFc1ccccc1\C=C\c1ccc2ccccc2n1
Structure
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