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TargetMucolipin-3
LigandBDBM46776
Substrate/Competitorn/a
Meas. Tech.Fluorescence counterscreen assay for TRPN1 agonists: dose response cell-based high-throughput screening assay to identify agonists of the transient receptor potential channel ML3 (TRPML3)
EC50 24300±n/a nM
Citation PubChem, PC Fluorescence counterscreen assay for TRPN1 agonists: dose response cell-based high-throughput screening assay to identify agonists of the transient receptor potential channel ML3 (TRPML3) PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Mucolipin-3
Name:Mucolipin-3
Synonyms:MCLN3_HUMAN | MCOLN3 | MCOLN3 protein
Type:Enzyme Catalytic Domain
Mol. Mass.:64244.09
Organism:Homo sapiens (Human)
Description:Q8TDD5
Residue:553
Sequence:
MADPEVVVSSCSSHEEENRCNFNQQTSPSEELLLEDQMRRKLKFFFMNPCEKFWARGRKP
WKLAIQILKIAMVTIQLVLFGLSNQMVVAFKEENTIAFKHLFLKGYMDRMDDTYAVYTQS
DVYDQLIFAVNQYLQLYNVSVGNHAYENKGTKQSAMAICQHFYKRGNIYPGNDTFDIDPE
IETECFFVEPDEPFHIGTPAENKLNLTLDFHRLLTVELQFKLKAINLQTVRHQELPDCYD
FTLTITFDNKAHSGRIKISLDNDISIRECKDWHVSGSIQKNTHYMMIFDAFVILTCLVSL
ILCIRSVIRGLQLQQEFVNFFLLHYKKEVSVSDQMEFVNGWYIMIIISDILTIIGSILKM
EIQAKSLTSYDVCSILLGTSTMLVWLGVIRYLGFFAKYNLLILTLQAALPNVIRFCCCAA
MIYLGYCFCGWIVLGPYHDKFRSLNMVSECLFSLINGDDMFATFAKMQQKSYLVWLFSRI
YLYSFISLFIYMILSLFIALITDTYETIKQYQQDGFPETELRTFISECKDLPNSGKYRLE
DDPPVSLFCCCKK
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  Blast E-value cutoff:
BDBM46776
n/a
NameBDBM46776
Synonyms:2-[(5-chloranylthiophen-2-yl)sulfonylamino]-N-[2-(phenylmethyl)phenyl]benzamide | 2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-[2-(phenylmethyl)phenyl]benzamide | MLS000401581 | N-(2-benzylphenyl)-2-[(5-chloro-2-thienyl)sulfonylamino]benzamide | N-(2-benzylphenyl)-2-[(5-chlorothiophen-2-yl)sulfonylamino]benzamide | SMR000243486 | cid_3677740
TypeSmall organic molecule
Emp. Form.C24H19ClN2O3S2
Mol. Mass.483.002
SMILESClc1ccc(s1)S(=O)(=O)Nc1ccccc1C(=O)Nc1ccccc1Cc1ccccc1
Structure
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