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TargetRegulator of G-protein signaling 4
LigandBDBM47700
Substrate/Competitorn/a
Meas. Tech.Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao.
EC50 30000±n/a nM
Citation PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Regulator of G-protein signaling 4
Name:Regulator of G-protein signaling 4
Synonyms:RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4)
Type:Enzyme
Mol. Mass.:23263.51
Organism:Homo sapiens (Human)
Description:P49798
Residue:205
Sequence:
MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47700
n/a
NameBDBM47700
Synonyms:2-(4-methyl-1-piperidinyl)aniline | 2-(4-methylpiperidin-1-yl)aniline | MLS000080408 | SMR000035930 | [2-(4-methylpiperidino)phenyl]amine | cid_663698
TypeSmall organic molecule
Emp. Form.C12H18N2
Mol. Mass.190.2847
SMILESCC1CCN(CC1)c1ccccc1N
Structure
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