| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 4 |
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| Ligand | BDBM47717 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. |
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| EC50 | 26420±n/a nM |
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| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Regulator of G-protein signaling 4 |
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| Name: | Regulator of G-protein signaling 4 |
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| Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 23263.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49798 |
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| Residue: | 205 |
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| Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
|
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|
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| BDBM47717 |
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| n/a |
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| Name | BDBM47717 |
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| Synonyms: | 5-Ethylamino-anthra[1,9-cd]isoxazol-6-one | MLS000525596 | SMR000116070 | cid_776361 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H12N2O2 |
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| Mol. Mass. | 264.2787 |
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| SMILES | CCNc1ccc2noc3-c4ccccc4C(=O)c1c23 |
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| Structure | 
|
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