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TargetRegulator of G-protein signaling 4
LigandBDBM47720
Substrate/Competitorn/a
Meas. Tech.Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao.
EC50 30000±n/a nM
Citation PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Regulator of G-protein signaling 4
Name:Regulator of G-protein signaling 4
Synonyms:RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4)
Type:Enzyme
Mol. Mass.:23263.51
Organism:Homo sapiens (Human)
Description:P49798
Residue:205
Sequence:
MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47720
n/a
NameBDBM47720
Synonyms:2-N,2-N-diethyl-4-N,4-N-diphenyl-1,3,5-triazine-2,4,6-triamine | MLS000522302 | N2,N2-diethyl-N4,N4-diphenyl-1,3,5-triazine-2,4,6-triamine | SMR000127570 | [4-amino-6-(diethylamino)-s-triazin-2-yl]-diphenyl-amine | cid_712290
TypeSmall organic molecule
Emp. Form.C19H22N6
Mol. Mass.334.4182
SMILESCCN(CC)c1nc(N)nc(n1)N(c1ccccc1)c1ccccc1
Structure
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