Reaction Details |
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Target | Regulator of G-protein signaling 4 |
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Ligand | BDBM47786 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. |
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EC50 | 30000±n/a nM |
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Citation | PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay(2009)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Regulator of G-protein signaling 4 |
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Name: | Regulator of G-protein signaling 4 |
Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
Type: | Enzyme |
Mol. Mass.: | 23263.51 |
Organism: | Homo sapiens (Human) |
Description: | P49798 |
Residue: | 205 |
Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47786 |
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n/a |
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Name | BDBM47786 |
Synonyms: | 6-chloro-3-pyridinecarboxylic acid [2-(tert-butylamino)-2-oxoethyl] ester | 6-chloronicotinic acid [2-(tert-butylamino)-2-keto-ethyl] ester | MLS000709523 | SMR000286890 | [2-(tert-butylamino)-2-oxidanylidene-ethyl] 6-chloranylpyridine-3-carboxylate | [2-(tert-butylamino)-2-oxoethyl] 6-chloropyridine-3-carboxylate | cid_2432404 |
Type | Small organic molecule |
Emp. Form. | C12H15ClN2O3 |
Mol. Mass. | 270.712 |
SMILES | CC(C)(C)NC(=O)COC(=O)c1ccc(Cl)nc1 |
Structure |
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