Reaction Details |
| Report a problem with these data |
Target | Dual specificity protein phosphatase 3 |
---|
Ligand | BDBM46229 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | Fluorescent assay for identification of compounds that inhibit VHR1 |
---|
IC50 | 1230±n/a nM |
---|
Citation | PubChem, PC Fluorescent assay for identification of compounds that inhibit VHR1 PubChem Bioassay(2009)[AID] |
---|
More Info.: | Get all data from this article, Solution Info, Assay Method |
---|
|
Dual specificity protein phosphatase 3 |
---|
Name: | Dual specificity protein phosphatase 3 |
Synonyms: | DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR |
Type: | Hydrolase |
Mol. Mass.: | 20480.58 |
Organism: | Homo sapiens (Human) |
Description: | n/a |
Residue: | 185 |
Sequence: | MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
|
|
|
BDBM46229 |
---|
n/a |
---|
Name | BDBM46229 |
Synonyms: | 4-chloranyl-N-(3,4-dihydro-2H-thiochromen-4-yl)-3-sulfamoyl-benzamide | 4-chloro-3-sulfamoyl-N-thiochroman-4-yl-benzamide | 4-chloro-N-(3,4-dihydro-2H-1-benzothiopyran-4-yl)-3-sulfamoylbenzamide | 4-chloro-N-(3,4-dihydro-2H-thiochromen-4-yl)-3-sulfamoylbenzamide | MLS-0336143.0001 | cid_16330874 |
Type | Small organic molecule |
Emp. Form. | C16H15ClN2O3S2 |
Mol. Mass. | 382.885 |
SMILES | NS(=O)(=O)c1cc(ccc1Cl)C(=O)NC1CCSc2ccccc12 |
Structure |
|