| Reaction Details |
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 | Report a problem with these data |
| Target | Dual specificity protein phosphatase 3 |
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| Ligand | BDBM46207 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescent assay for identification of compounds that inhibit VHR1 |
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| IC50 | 1880±n/a nM |
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| Citation |  PubChem, PC Fluorescent assay for identification of compounds that inhibit VHR1 PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Dual specificity protein phosphatase 3 |
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| Name: | Dual specificity protein phosphatase 3 |
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| Synonyms: | DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR |
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| Type: | Hydrolase |
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| Mol. Mass.: | 20480.58 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 185 |
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| Sequence: | MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
|
|
|
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| BDBM46207 |
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| n/a |
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| Name | BDBM46207 |
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| Synonyms: | 4-[[5-(4-bromophenyl)-2-furoyl]thiocarbamoylamino]benzoic acid | 4-[[5-(4-bromophenyl)furan-2-carbonyl]carbamothioylamino]benzoic acid | 4-[[5-(4-bromophenyl)furan-2-yl]carbonylcarbamothioylamino]benzoic acid | 4-[[[[[5-(4-bromophenyl)-2-furanyl]-oxomethyl]amino]-sulfanylidenemethyl]amino]benzoic acid | MLS-0383777.0001 | cid_1328767 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H13BrN2O4S |
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| Mol. Mass. | 445.287 |
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| SMILES | OC(=O)c1ccc(NC(=S)NC(=O)c2ccc(o2)-c2ccc(Br)cc2)cc1 |
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| Structure | 
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