Ki Summary

Reaction Details

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Target

Zinc finger protein mex-5

Ligand

BDBM52500

Substrate/Competitor

n/a

Meas. Tech.

Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2

EC50

300000±n/a nM

Citation

PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Zinc finger protein mex-5

Name:

Zinc finger protein mex-5

Synonyms:

MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5

Type:

Enzyme Catalytic Domain

Mol. Mass.:

52832.78

Organism:

Caenorhabditis elegans

Description:

gi_55976631

Residue:

468

Sequence:

MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNG
SSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQP
QLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTA
PLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAE
KENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKE
LRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDD
QDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGD
YNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY

BDBM52500

n/a

Name

BDBM52500

Synonyms:

3-(4-fluorophenyl)-1-phenyl-4-pyrazolecarboxylic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] ester | 3-(4-fluorophenyl)-1-phenyl-pyrazole-4-carboxylic acid [2-keto-2-(4-sulfamoylanilino)ethyl] ester | MLS000374593 | SMR000244208 | [2-oxidanylidene-2-[(4-sulfamoylphenyl)amino]ethyl] 3-(4-fluorophenyl)-1-phenyl-pyrazole-4-carboxylate | [2-oxo-2-(4-sulfamoylanilino)ethyl] 3-(4-fluorophenyl)-1-phenylpyrazole-4-carboxylate | cid_2379848

Type

Small organic molecule

Emp. Form.

C24H19FN4O5S

Mol. Mass.

494.495

SMILES

NS(=O)(=O)c1ccc(NC(=O)COC(=O)c2cn(nc2-c2ccc(F)cc2)-c2ccccc2)cc1

Structure