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TargetPOsterior Segregation
LigandBDBM52869
Substrate/Competitorn/a
Meas. Tech.Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50 7981±n/a nM
Citation PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
POsterior Segregation
Name:POsterior Segregation
Synonyms:POsterior Segregation family member (pos-1)
Type:Enzyme Catalytic Domain
Mol. Mass.:29838.90
Organism:Caenorhabditis elegans
Description:gi_17562800
Residue:264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKET
QNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCR
FAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGA
HANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYN
STAQLAQYFESQFQRIQQLSSHHH
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BDBM52869
n/a
NameBDBM52869
Synonyms:5-[2-[(E)-(3-methoxy-5-nitro-4-oxidanylidene-cyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]-6-methyl-2H-1,2,4-triazin-3-one | 5-[2-[(E)-(3-methoxy-5-nitro-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]-6-methyl-2H-1,2,4-triazin-3-one | 5-[N'-[(E)-(4-keto-3-methoxy-5-nitro-cyclohexa-2,5-dien-1-ylidene)methyl]hydrazino]-6-methyl-2H-1,2,4-triazin-3-one | 5-[[(E)-(3-methoxy-5-nitro-4-oxo-1-cyclohexa-2,5-dienylidene)methyl]hydrazo]-6-methyl-2H-1,2,4-triazin-3-one | 5-{N'-[1-(4-Hydroxy-3-methoxy-5-nitro-phenyl)-meth-(E)-ylidene]-hydrazino}-6-methyl-2H-[1,2,4]triazin-3- one | MLS000777029 | SMR000413418 | cid_5710929
TypeSmall organic molecule
Emp. Form.C12H12N6O5
Mol. Mass.320.2609
SMILESCOc1c[c-](C[NH+]=Nc2[nH]c(=O)nnc2C)cc([N+]([O-])=O)c1=O |w:6.5|
Structure
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