| Reaction Details |
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 | Report a problem with these data |
| Target | POsterior Segregation |
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| Ligand | BDBM52465 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA |
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| EC50 | 103696±n/a nM |
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| Citation |  PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| POsterior Segregation |
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| Name: | POsterior Segregation |
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| Synonyms: | POsterior Segregation family member (pos-1) |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 29838.90 |
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| Organism: | Caenorhabditis elegans |
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| Description: | gi_17562800 |
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| Residue: | 264 |
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| Sequence: | MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKET
QNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCR
FAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGA
HANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYN
STAQLAQYFESQFQRIQQLSSHHH
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| BDBM52465 |
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| n/a |
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| Name | BDBM52465 |
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| Synonyms: | (E)-2-Cyano-3-[2-(3,5-dimethyl-phenoxy)-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]-acrylic acid methyl ester | (E)-2-cyano-3-[2-(3,5-dimethylphenoxy)-4-keto-9-methyl-pyrido[1,2-a]pyrimidin-3-yl]acrylic acid methyl ester | (E)-2-cyano-3-[2-(3,5-dimethylphenoxy)-9-methyl-4-oxo-3-pyrido[1,2-a]pyrimidinyl]-2-propenoic acid methyl ester | MLS000588134 | SMR000220196 | cid_2017737 | methyl (E)-2-cyano-3-[2-(3,5-dimethylphenoxy)-9-methyl-4-oxidanylidene-pyrido[1,2-a]pyrimidin-3-yl]prop-2-enoate | methyl (E)-2-cyano-3-[2-(3,5-dimethylphenoxy)-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enoate |
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| Type | Small organic molecule |
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| Emp. Form. | C22H19N3O4 |
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| Mol. Mass. | 389.404 |
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| SMILES | COC(=O)C(=C\c1c(Oc2cc(C)cc(C)c2)nc2c(C)cccn2c1=O)\C#N |
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| Structure | 
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