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TargetPOsterior Segregation
LigandBDBM52482
Substrate/Competitorn/a
Meas. Tech.Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50 300000±n/a nM
Citation PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
POsterior Segregation
Name:POsterior Segregation
Synonyms:POsterior Segregation family member (pos-1)
Type:Enzyme Catalytic Domain
Mol. Mass.:29838.90
Organism:Caenorhabditis elegans
Description:gi_17562800
Residue:264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKET
QNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCR
FAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGA
HANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYN
STAQLAQYFESQFQRIQQLSSHHH
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BDBM52482
n/a
NameBDBM52482
Synonyms:4-[2,5-dimethyl-3-[2-[2-(tosylamino)acetyl]oxyacetyl]pyrrol-1-yl]benzoic acid methyl ester | 4-[2,5-dimethyl-3-[2-[2-[(4-methylphenyl)sulfonylamino]-1-oxoethoxy]-1-oxoethyl]-1-pyrrolyl]benzoic acid methyl ester | MLS000393606 | SMR000247827 | cid_2127943 | methyl 4-[2,5-dimethyl-3-[2-[2-[(4-methylphenyl)sulfonylamino]acetyl]oxyacetyl]pyrrol-1-yl]benzoate | methyl 4-[2,5-dimethyl-3-[2-[2-[(4-methylphenyl)sulfonylamino]ethanoyloxy]ethanoyl]pyrrol-1-yl]benzoate
TypeSmall organic molecule
Emp. Form.C25H26N2O7S
Mol. Mass.498.548
SMILESCOC(=O)c1ccc(cc1)-n1c(C)cc(C(=O)COC(=O)CNS(=O)(=O)c2ccc(C)cc2)c1C
Structure
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