| Reaction Details |
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 | Report a problem with these data |
| Target | SUMO-conjugating enzyme UBC9 |
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| Ligand | BDBM61233 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | AlphaScreen confirmatory assay for validation of inhibitors of SUMOylation |
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| IC50 | 2110±n/a nM |
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| Citation |  PubChem, PC AlphaScreen confirmatory assay for validation of inhibitors of SUMOylation PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| SUMO-conjugating enzyme UBC9 |
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| Name: | SUMO-conjugating enzyme UBC9 |
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| Synonyms: | UBC9 | UBC9_HUMAN | UBCE9 | UBE2I | ubiquitin-conjugating enzyme E2I |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 18011.66 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_4507785 |
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| Residue: | 158 |
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| Sequence: | MSGIALSRLAQERKAWRKDHPFGFVAVPTKNPDGTMNLMNWECAIPGKKGTPWEGGLFKL
RMLFKDDYPSSPPKCKFEPPLFHPNVYPSGTVCLSILEEDKDWRPAITIKQILLGIQELL
NEPNIQDPAQAEAYTIYCQNRVEYEKRVRAQAKKFAPS
|
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| BDBM61233 |
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| n/a |
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| Name | BDBM61233 |
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| Synonyms: | 4-[(3,4-diketo-1-naphthyl)amino]benzenesulfonamide | 4-[(3,4-dioxo-1-naphthalenyl)amino]benzenesulfonamide | 4-[(3,4-dioxo-3,4-dihydro-1-naphthalenyl)amino]benzenesulfonamide | 4-[(3,4-dioxonaphthalen-1-yl)amino]benzenesulfonamide | 4-[[3,4-bis(oxidanylidene)naphthalen-1-yl]amino]benzenesulfonamide | MLS001164435 | SMR000496650 | cid_367783 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H12N2O4S |
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| Mol. Mass. | 328.342 |
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| SMILES | NS(=O)(=O)c1ccc(NC2=CC(=O)C(=O)c3ccccc23)cc1 |t:9| |
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| Structure | 
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