| Reaction Details |
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 | Report a problem with these data |
| Target | SUMO-conjugating enzyme UBC9 |
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| Ligand | BDBM53205 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | AlphaScreen confirmatory assay for validation of inhibitors of SUMOylation |
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| IC50 | 690±n/a nM |
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| Citation |  PubChem, PC AlphaScreen confirmatory assay for validation of inhibitors of SUMOylation PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| SUMO-conjugating enzyme UBC9 |
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| Name: | SUMO-conjugating enzyme UBC9 |
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| Synonyms: | UBC9 | UBC9_HUMAN | UBCE9 | UBE2I | ubiquitin-conjugating enzyme E2I |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 18011.66 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_4507785 |
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| Residue: | 158 |
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| Sequence: | MSGIALSRLAQERKAWRKDHPFGFVAVPTKNPDGTMNLMNWECAIPGKKGTPWEGGLFKL
RMLFKDDYPSSPPKCKFEPPLFHPNVYPSGTVCLSILEEDKDWRPAITIKQILLGIQELL
NEPNIQDPAQAEAYTIYCQNRVEYEKRVRAQAKKFAPS
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| BDBM53205 |
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| n/a |
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| Name | BDBM53205 |
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| Synonyms: | 1,3-bis[[(Z)-(3-hydroxy-4-keto-cyclohexa-2,5-dien-1-ylidene)methyl]amino]urea | 1,3-bis[[(Z)-(3-hydroxy-4-oxo-1-cyclohexa-2,5-dienylidene)methyl]amino]urea | 1,3-bis[[(Z)-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]amino]urea | 1,3-bis[[(Z)-(3-oxidanyl-4-oxidanylidene-cyclohexa-2,5-dien-1-ylidene)methyl]amino]urea | MLS001202140 | N'',N'''-bis[(1E)-(3,4-dihydroxyphenyl)methylene]carbonohydrazide | SMR000565039 | cid_24762014 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H14N4O5 |
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| Mol. Mass. | 330.2955 |
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| SMILES | O=C(NN=CC1=CC(=O)C(=O)CC1)NN=CC1=CC(=O)C(=O)CC1 |w:3.2,14.14,t:5,17| |
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| Structure | 
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