| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cell division control protein 42 homolog |
|---|
| Ligand | BDBM54596 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 wildtype protein |
|---|
| EC50 | 30000±n/a nM |
|---|
| Citation |  PubChem, PC Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 wildtype protein PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Cell division control protein 42 homolog |
|---|
| Name: | Cell division control protein 42 homolog |
|---|
| Synonyms: | CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa) |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 21258.36 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_652970 |
|---|
| Residue: | 191 |
|---|
| Sequence: | MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
|
|
|
|---|
| BDBM54596 |
|---|
| n/a |
|---|
| Name | BDBM54596 |
|---|
| Synonyms: | UNM-0000305834 | cid_23669604 | sodium;4-(3,5-diphenyl-2-pyrazolin-1-yl)besylate | sodium;4-(3,5-diphenyl-3,4-dihydropyrazol-2-yl)benzenesulfonate |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H17N2O3S |
|---|
| Mol. Mass. | 377.437 |
|---|
| SMILES | [O-]S(=O)(=O)c1ccc(cc1)N1N=C(CC1c1ccccc1)c1ccccc1 |c:12| |
|---|
| Structure | 
|
|---|
Search and Browse
