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TargetCell division control protein 42 homolog
LigandBDBM54677
Substrate/Competitorn/a
Meas. Tech.Additional SAR compounds tested by Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant
EC50 30000±n/a nM
Citation PubChem, PC Additional SAR compounds tested by Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cell division control protein 42 homolog
Name:Cell division control protein 42 homolog
Synonyms:CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa)
Type:PROTEIN
Mol. Mass.:21258.36
Organism:Homo sapiens (Human)
Description:ChEMBL_652970
Residue:191
Sequence:
MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
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BDBM54677
n/a
NameBDBM54677
Synonyms:(3E)-3-(1-ketoindan-2-ylidene)oxindole | (3E)-3-(3-oxidanylidene-1H-inden-2-ylidene)-1H-indol-2-one | (3E)-3-(3-oxo-1H-inden-2-ylidene)-1H-indol-2-one | UNM-0000305763 | cid_25220924
TypeSmall organic molecule
Emp. Form.C17H11NO2
Mol. Mass.261.2747
SMILESO=C1Nc2ccccc2\C1=C1\Cc2ccccc2C1=O
Structure
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