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TargetCell division control protein 42 homolog
LigandBDBM54694
Substrate/Competitorn/a
Meas. Tech.Additional SAR compounds tested by Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant
EC50 30000±n/a nM
Citation PubChem, PC Additional SAR compounds tested by Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cell division control protein 42 homolog
Name:Cell division control protein 42 homolog
Synonyms:CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa)
Type:PROTEIN
Mol. Mass.:21258.36
Organism:Homo sapiens (Human)
Description:ChEMBL_652970
Residue:191
Sequence:
MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
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BDBM54694
n/a
NameBDBM54694
Synonyms:1-(2-nitrophenyl)-3-phenyl-2-propyn-1-one | 1-(2-nitrophenyl)-3-phenyl-prop-2-yn-1-one | 1-(2-nitrophenyl)-3-phenylprop-2-yn-1-one | UNM-0000306038 | cid_25227393
TypeSmall organic molecule
Emp. Form.C15H9NO3
Mol. Mass.251.2369
SMILES[O-][N+](=O)c1ccccc1C(=O)C#Cc1ccccc1
Structure
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