| Reaction Details |
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 | Report a problem with these data |
| Target | Ras-related C3 botulinum toxin substrate 1 |
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| Ligand | BDBM54676 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype |
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| EC50 | 1667±n/a nM |
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| Citation |  PubChem, PC Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Ras-related C3 botulinum toxin substrate 1 |
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| Name: | Ras-related C3 botulinum toxin substrate 1 |
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| Synonyms: | RAC1_MOUSE | Rac1 | Rac1 protein |
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| Type: | PROTEIN |
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| Mol. Mass.: | 21455.91 |
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| Organism: | Mus musculus |
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| Description: | EBI_101485 |
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| Residue: | 192 |
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| Sequence: | MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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| BDBM54676 |
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| n/a |
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| Name | BDBM54676 |
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| Synonyms: | (3Z)-3-(5-keto-2-thioxo-imidazolidin-4-ylidene)oxindole | (3Z)-3-(5-oxidanylidene-2-sulfanylidene-imidazolidin-4-ylidene)-1H-indol-2-one | (3Z)-3-(5-oxo-2-sulfanylidene-4-imidazolidinylidene)-1H-indol-2-one | (3Z)-3-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)-1H-indol-2-one | UNM-0000305762 | cid_5339891 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H7N3O2S |
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| Mol. Mass. | 245.257 |
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| SMILES | O=C1NC(=S)N\C1=C1/C(=O)Nc2ccccc12 |
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| Structure | 
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