| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Ras-related C3 botulinum toxin substrate 1 |
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| Ligand | BDBM54678 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype |
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| EC50 | 30000±n/a nM |
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| Citation |  PubChem, PC Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Ras-related C3 botulinum toxin substrate 1 |
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| Name: | Ras-related C3 botulinum toxin substrate 1 |
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| Synonyms: | RAC1_MOUSE | Rac1 | Rac1 protein |
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| Type: | PROTEIN |
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| Mol. Mass.: | 21455.91 |
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| Organism: | Mus musculus |
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| Description: | EBI_101485 |
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| Residue: | 192 |
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| Sequence: | MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
|
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|
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| BDBM54678 |
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| n/a |
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| Name | BDBM54678 |
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| Synonyms: | (3E)-7-bromanyl-3-(3-oxidanylidene-1H-inden-2-ylidene)-1H-indol-2-one | (3E)-7-bromo-3-(1-ketoindan-2-ylidene)oxindole | (3E)-7-bromo-3-(3-oxo-1H-inden-2-ylidene)-1H-indol-2-one | UNM-0000305764 | cid_25220925 |
|---|
| Type | Small organic molecule |
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| Emp. Form. | C17H10BrNO2 |
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| Mol. Mass. | 340.171 |
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| SMILES | Brc1cccc2\C(C(=O)Nc12)=C1\Cc2ccccc2C1=O |
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| Structure | 
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