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TargetRas-related C3 botulinum toxin substrate 1
LigandBDBM50218896
Substrate/Competitorn/a
Meas. Tech.Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype
EC50 34594±n/a nM
Citation PubChem, PC Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Ras-related C3 botulinum toxin substrate 1
Name:Ras-related C3 botulinum toxin substrate 1
Synonyms:RAC1_MOUSE | Rac1 | Rac1 protein
Type:PROTEIN
Mol. Mass.:21455.91
Organism:Mus musculus
Description:EBI_101485
Residue:192
Sequence:
MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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  Blast E-value cutoff:
BDBM50218896
n/a
NameBDBM50218896
Synonyms:7-fluoroindirubin | CHEMBL243986 | cid_11847138
TypeSmall organic molecule
Emp. Form.C16H9FN2O2
Mol. Mass.280.2533
SMILESFc1cccc2C(C(=O)Nc12)=C1Nc2ccccc2C1=O |w:11.13|
Structure
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