| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Ras-related C3 botulinum toxin substrate 1 |
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| Ligand | BDBM54683 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype |
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| EC50 | 30000±n/a nM |
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| Citation |  PubChem, PC Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Ras-related C3 botulinum toxin substrate 1 |
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| Name: | Ras-related C3 botulinum toxin substrate 1 |
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| Synonyms: | RAC1_MOUSE | Rac1 | Rac1 protein |
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| Type: | PROTEIN |
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| Mol. Mass.: | 21455.91 |
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| Organism: | Mus musculus |
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| Description: | EBI_101485 |
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| Residue: | 192 |
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| Sequence: | MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
|
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|
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| BDBM54683 |
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| n/a |
|---|
| Name | BDBM54683 |
|---|
| Synonyms: | 7-fluoranyl-3-[3-(oxidanylamino)-1H-indol-2-yl]indol-2-one | 7-fluoro-3-[3-(hydroxyamino)-1H-indol-2-yl]-2-indolone | 7-fluoro-3-[3-(hydroxyamino)-1H-indol-2-yl]indol-2-one | UNM-0000305773 | cid_11845975 |
|---|
| Type | Small organic molecule |
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| Emp. Form. | C16H10FN3O2 |
|---|
| Mol. Mass. | 295.2679 |
|---|
| SMILES | ONc1c([nH]c2ccccc12)C1=c2cccc(F)c2=NC1=O |c:13,21| |
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| Structure | 
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