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TargetRas-related C3 botulinum toxin substrate 1
LigandBDBM54699
Substrate/Competitorn/a
Meas. Tech.Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype
EC50 30000±n/a nM
Citation PubChem, PC Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Ras-related C3 botulinum toxin substrate 1
Name:Ras-related C3 botulinum toxin substrate 1
Synonyms:RAC1_MOUSE | Rac1 | Rac1 protein
Type:PROTEIN
Mol. Mass.:21455.91
Organism:Mus musculus
Description:EBI_101485
Residue:192
Sequence:
MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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BDBM54699
n/a
NameBDBM54699
Synonyms:4-(1-oxo-3-phenylprop-2-ynyl)benzonitrile | 4-(3-phenylprop-2-ynoyl)benzenecarbonitrile | 4-(3-phenylprop-2-ynoyl)benzonitrile | 4-(3-phenylpropioloyl)benzonitrile | UNM-0000306057 | cid_11708441
TypeSmall organic molecule
Emp. Form.C16H9NO
Mol. Mass.231.2488
SMILESO=C(C#Cc1ccccc1)c1ccc(cc1)C#N
Structure
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