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TargetRas-related protein Rab-2A
LigandBDBM54694
Substrate/Competitorn/a
Meas. Tech.Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rab2 wildtype
EC50 30000±n/a nM
Citation PubChem, PC Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rab2 wildtype PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Ras-related protein Rab-2A
Name:Ras-related protein Rab-2A
Synonyms:RAB2 | RAB2A | RAB2A_CANLF | Ras-related protein Rab-2A.
Type:Enzyme Catalytic Domain
Mol. Mass.:23545.28
Organism:Canis lupus familiaris
Description:gi_46577642
Residue:212
Sequence:
MAYAYLFKYIIIGDTGVGKSCLLLQFTDKRFQPVHDLTIGVEFGARMITIDGKQIKLQIW
DTAGQESFRSITRSYYRGAAGALLVYDITRRDTFNHLTTWLEDARQHSNSNMVIMLIGNK
SDLESRREVKKEEGEAFAREHGLIFMETSAKTASNVEEAFINTAKEIYEKIQEGVFDINN
EANGIKIGPQHAATNATHAGNQGGQQAGGGCC
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  Blast E-value cutoff:
BDBM54694
n/a
NameBDBM54694
Synonyms:1-(2-nitrophenyl)-3-phenyl-2-propyn-1-one | 1-(2-nitrophenyl)-3-phenyl-prop-2-yn-1-one | 1-(2-nitrophenyl)-3-phenylprop-2-yn-1-one | UNM-0000306038 | cid_25227393
TypeSmall organic molecule
Emp. Form.C15H9NO3
Mol. Mass.251.2369
SMILES[O-][N+](=O)c1ccccc1C(=O)C#Cc1ccccc1
Structure
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