| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Ras-related C3 botulinum toxin substrate 1 |
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| Ligand | BDBM13063 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype |
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| EC50 | 30000±n/a nM |
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| Citation |  PubChem, PC Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Ras-related C3 botulinum toxin substrate 1 |
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| Name: | Ras-related C3 botulinum toxin substrate 1 |
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| Synonyms: | RAC1_MOUSE | Rac1 | Rac1 protein |
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| Type: | PROTEIN |
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| Mol. Mass.: | 21455.91 |
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| Organism: | Mus musculus |
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| Description: | EBI_101485 |
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| Residue: | 192 |
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| Sequence: | MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
|
|
|
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| BDBM13063 |
|---|
| n/a |
|---|
| Name | BDBM13063 |
|---|
| Synonyms: | 4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)benzene-1-sulfonamide | Bextra | CHEMBL865 | VLX | Valdecoxib | cid_119607 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H14N2O3S |
|---|
| Mol. Mass. | 314.359 |
|---|
| SMILES | Cc1onc(c1-c1ccc(cc1)S(N)(=O)=O)-c1ccccc1 |
|---|
| Structure | 
|
|---|
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