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Reaction Details
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TargetRas-related C3 botulinum toxin substrate 1
LigandBDBM54616
Substrate/Competitorn/a
Meas. Tech.Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype
EC50 30000±n/a nM
Citation PubChem, PC Pyrazoline SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Ras-related C3 botulinum toxin substrate 1
Name:Ras-related C3 botulinum toxin substrate 1
Synonyms:RAC1_MOUSE | Rac1 | Rac1 protein
Type:PROTEIN
Mol. Mass.:21455.91
Organism:Mus musculus
Description:EBI_101485
Residue:192
Sequence:
MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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  Blast E-value cutoff:
BDBM54616
n/a
NameBDBM54616
Synonyms:1-(2-methoxyphenyl)-3,5-diphenyl-2-pyrazoline | 2-(2-methoxyphenyl)-3,5-diphenyl-3,4-dihydropyrazole | UNM-0000305855 | cid_2865685
TypeSmall organic molecule
Emp. Form.C22H20N2O
Mol. Mass.328.407
SMILESCOc1ccccc1N1N=C(CC1c1ccccc1)c1ccccc1 |c:10|
Structure
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