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TargetBcl-2-related protein A1
LigandBDBM33111
Substrate/Competitorn/a
Meas. Tech.Confirmation dose response of hits from multiplexed high-throughput screen for small molecule regulators of Bcl-2 family protein interactions, specifically Bim-Bfl-1
EC50 3970±n/a nM
Citation PubChem, PC Confirmation dose response of hits from multiplexed high-throughput screen for small molecule regulators of Bcl-2 family protein interactions, specifically Bim-Bfl-1 PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Bcl-2-related protein A1
Name:Bcl-2-related protein A1
Synonyms:B2LA1_HUMAN | BCL2A1 | BCL2L5 | BFL1 | Bcl-2-like protein 5 | GRS | HBPA1 | Hemopoietic-specific early response protein | Protein BFL-1 | Protein GRS
Type:Apoptosis regulator protein
Mol. Mass.:20130.01
Organism:Homo sapiens (Human)
Description:n/a
Residue:175
Sequence:
MTDCEFGYIYRLAQDYLQCVLQIPQPGSGPSKTSRVLQNVAFSVQKEVEKNLKSCLDNVN
VVSVDTARTLFNQVMEKEFEDGIINWGRIVTIFAFEGILIKKLLRQQIAPDVDTYKEISY
FVAEFIMNNTGEWIRQNGGWENGFVKKFEPKSGWMTFLEVTGKICEMLSLLKQYC
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BDBM33111
n/a
NameBDBM33111
Synonyms:4,4,4-Trichloro-3-methylamino-1-(4-nitro-phenyl)-butan-1-one | 4,4,4-trichloro-3-(methylamino)-1-(4-nitrophenyl)-1-butanone | 4,4,4-trichloro-3-(methylamino)-1-(4-nitrophenyl)butan-1-one | 4,4,4-tris(chloranyl)-3-(methylamino)-1-(4-nitrophenyl)butan-1-one | MLS000590271 | SMR000217256 | cid_3739292
TypeSmall organic molecule
Emp. Form.C11H11Cl3N2O3
Mol. Mass.325.576
SMILESCNC(CC(=O)c1ccc(cc1)[N+]([O-])=O)C(Cl)(Cl)Cl
Structure
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