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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Metabotropic glutamate receptor 4 [Q124R] | ||
| Ligand | BDBM55091 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Modulation of the Metabotropic Glutamate Receptor mGluR4: Rat PAM Potency | ||
| EC50 | 690±n/a nM | ||
| Citation |  PubChem, PC Modulation of the Metabotropic Glutamate Receptor mGluR4: Rat PAM Potency PubChem Bioassay(2010)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| Metabotropic glutamate receptor 4 [Q124R] | |||
| Name: | Metabotropic glutamate receptor 4 [Q124R] | ||
| Synonyms: | GRM4_RAT | Gprc1d | Grm4 | Mglur4 | glutamate receptor, metabotropic 4 precursor | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 101878.86 | ||
| Organism: | Rattus norvegicus | ||
| Description: | gi_12083595 | ||
| Residue: | 912 | ||
| Sequence: |
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| BDBM55091 | |||
| n/a | |||
| Name | BDBM55091 | ||
| Synonyms: | N-[3-chloranyl-4-[(1S,5R)-6,6-dimethyl-2,4-bis(oxidanylidene)-3-azabicyclo[3.1.0]hexan-3-yl]phenyl]pyridine-2-carboxamide | N-[3-chloro-4-[(1S,5R)-2,4-diketo-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-3-yl]phenyl]picolinamide | N-[3-chloro-4-[(1S,5R)-6,6-dimethyl-2,4-dioxo-3-azabicyclo[3.1.0]hexan-3-yl]phenyl]-2-pyridinecarboxamide | N-[3-chloro-4-[(1S,5R)-6,6-dimethyl-2,4-dioxo-3-azabicyclo[3.1.0]hexan-3-yl]phenyl]pyridine-2-carboxamide | VU0410425-1 | cid_46869949 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C19H16ClN3O3 | ||
| Mol. Mass. | 369.802 | ||
| SMILES | CC1(C)c2c1c(O)n(c2O)-c1ccc(NC(=O)c2ccccn2)cc1Cl |(19.1,-1.33,;18.33,,;19.1,1.33,;17,.77,;17,-.77,;15.54,-1.25,;15.06,-2.71,;14.63,,;15.54,1.25,;15.06,2.71,;13.09,,;12.32,-1.33,;10.78,-1.33,;10.01,,;8.47,,;7.7,-1.33,;8.47,-2.67,;6.16,-1.33,;5.39,,;3.85,,;3.08,-1.33,;3.85,-2.67,;5.39,-2.67,;10.78,1.33,;12.32,1.33,;13.09,2.67,)| | ||
| Structure | 
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