| Reaction Details |
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 | Report a problem with these data |
| Target | M18 aspartyl aminopeptidase |
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| Ligand | BDBM55117 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | QFRET-based biochemical high throughput dose response assay for inhibitors of the Plasmodium falciparum M18 Aspartyl Aminopeptidase (PFM18AAP). |
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| IC50 | 497.28±n/a nM |
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| Citation |  PubChem, PC QFRET-based biochemical high throughput dose response assay for inhibitors of the Plasmodium falciparum M18 Aspartyl Aminopeptidase (PFM18AAP). PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| M18 aspartyl aminopeptidase |
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| Name: | M18 aspartyl aminopeptidase |
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| Synonyms: | n/a |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 65642.43 |
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| Organism: | Plasmodium falciparum 3D7 |
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| Description: | gi_23505220 |
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| Residue: | 570 |
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| Sequence: | MDKKAREYAQDALKFIQRSGSNFLACKNLKERLENNGFINLSEGETWNLNKNEGYVLCKE
NRNICGFFVGKNFNIDTGSILISIGHIDSCALKISPNNNVIKKKIHQINVECYGSGLWHT
WFDRSLGLSGQVLYKKGNKLVEKLIQINKSVLFLPSLAIHLQNRTRYDFSVKINYENHIK
PIISTTLFNQLNKCKRNNVHHDTILTTDTKFSHKENSQNKRDDQMCHSFNDKDVSNHNLD
KNTIEHLTNQQNEEKNKHTKDNPNSKDIVEHINTDNSYPLLYLLSKELNCKEEDILDFEL
CLMDTQEPCFTGVYEEFIEGARFDNLLGSFCVFEGFIELVNSIKNHTSNENTNHTNNITN
DINDNIHNNLYISIGYDHEEIGSLSEVGARSYCTKNFIDRIISSVFKKEIHEKNLSVQEI
YGNLVNRSFILNVDMAHCSHPNYPETVQDNHQLFFHEGIAIKYNTNKNYVTSPLHASLIK
RTFELYYNKYKQQIKYQNFMVKNDTPCGSTVGSMVAANLSMPGIDIGIPQLAMHSIREIA
AVHDVFFLIKGVFAFYTYYNQVLSTCVHDK
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| BDBM55117 |
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| n/a |
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| Name | BDBM55117 |
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| Synonyms: | 2-[benzenesulfonyl(1,2,4-triazol-4-yl)amino]acetic acid methyl ester | 2-[besyl(1,2,4-triazol-4-yl)amino]acetic acid methyl ester | MLS000111921 | SMR000107840 | cid_805790 | methyl 2-[benzenesulfonyl(1,2,4-triazol-4-yl)amino]acetate | methyl 2-[phenylsulfonyl(1,2,4-triazol-4-yl)amino]ethanoate |
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| Type | Small organic molecule |
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| Emp. Form. | C11H12N4O4S |
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| Mol. Mass. | 296.302 |
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| SMILES | COC(=O)CN(n1cnnc1)S(=O)(=O)c1ccccc1 |
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| Structure | 
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