| Reaction Details |
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 | Report a problem with these data |
| Target | M18 aspartyl aminopeptidase |
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| Ligand | BDBM55154 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | QFRET-based biochemical high throughput dose response assay for inhibitors of the Plasmodium falciparum M18 Aspartyl Aminopeptidase (PFM18AAP). |
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| IC50 | >100.76±n/a nM |
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| Citation |  PubChem, PC QFRET-based biochemical high throughput dose response assay for inhibitors of the Plasmodium falciparum M18 Aspartyl Aminopeptidase (PFM18AAP). PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| M18 aspartyl aminopeptidase |
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| Name: | M18 aspartyl aminopeptidase |
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| Synonyms: | n/a |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 65642.43 |
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| Organism: | Plasmodium falciparum 3D7 |
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| Description: | gi_23505220 |
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| Residue: | 570 |
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| Sequence: | MDKKAREYAQDALKFIQRSGSNFLACKNLKERLENNGFINLSEGETWNLNKNEGYVLCKE
NRNICGFFVGKNFNIDTGSILISIGHIDSCALKISPNNNVIKKKIHQINVECYGSGLWHT
WFDRSLGLSGQVLYKKGNKLVEKLIQINKSVLFLPSLAIHLQNRTRYDFSVKINYENHIK
PIISTTLFNQLNKCKRNNVHHDTILTTDTKFSHKENSQNKRDDQMCHSFNDKDVSNHNLD
KNTIEHLTNQQNEEKNKHTKDNPNSKDIVEHINTDNSYPLLYLLSKELNCKEEDILDFEL
CLMDTQEPCFTGVYEEFIEGARFDNLLGSFCVFEGFIELVNSIKNHTSNENTNHTNNITN
DINDNIHNNLYISIGYDHEEIGSLSEVGARSYCTKNFIDRIISSVFKKEIHEKNLSVQEI
YGNLVNRSFILNVDMAHCSHPNYPETVQDNHQLFFHEGIAIKYNTNKNYVTSPLHASLIK
RTFELYYNKYKQQIKYQNFMVKNDTPCGSTVGSMVAANLSMPGIDIGIPQLAMHSIREIA
AVHDVFFLIKGVFAFYTYYNQVLSTCVHDK
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| BDBM55154 |
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| n/a |
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| Name | BDBM55154 |
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| Synonyms: | 2-benzyl-4,6-dinitro-1,2-benzisothiazol-3(2H)-one | 2-benzyl-4,6-dinitro-1,2-benzothiazol-3-one | 4,6-dinitro-2-(phenylmethyl)-1,2-benzothiazol-3-one | MLS001198480 | SMR000559116 | cid_4652205 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H9N3O5S |
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| Mol. Mass. | 331.303 |
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| SMILES | [O-][N+](=O)c1cc([N+]([O-])=O)c2c(c1)sn(Cc1ccccc1)c2=O |
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| Structure | 
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