| Reaction Details |
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 | Report a problem with these data |
| Target | Kallikrein-5 |
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| Ligand | BDBM56239 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Kallikrein 5 1536 HTS Dose Response Confirmation |
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| IC50 | 2425.41±n/a nM |
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| Citation |  PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Kallikrein-5 |
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| Name: | Kallikrein-5 |
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| Synonyms: | KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein |
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| Type: | PROTEIN |
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| Mol. Mass.: | 32031.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | EBI_12584 |
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| Residue: | 293 |
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| Sequence: | MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARS
DDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGH
YSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPS
AGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDS
CQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
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| BDBM56239 |
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| n/a |
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| Name | BDBM56239 |
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| Synonyms: | 1-(3,5-dimethyl-1-thiophen-2-ylcarbonyl-pyrazol-4-yl)ethanone | 1-[3,5-dimethyl-1-(2-thenoyl)pyrazol-4-yl]ethanone | 1-[3,5-dimethyl-1-(thiophene-2-carbonyl)pyrazol-4-yl]ethanone | 1-[3,5-dimethyl-1-[oxo(thiophen-2-yl)methyl]-4-pyrazolyl]ethanone | MLS000115869 | SMR000092877 | cid_712603 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H12N2O2S |
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| Mol. Mass. | 248.301 |
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| SMILES | CC(=O)c1c(C)nn(C(=O)c2cccs2)c1C |
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| Structure | 
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