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TargetKallikrein-5
LigandBDBM33449
Substrate/Competitorn/a
Meas. Tech.Kallikrein 5 1536 HTS Dose Response Confirmation
IC50 1937.29±n/a nM
Citation PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Kallikrein-5
Name:Kallikrein-5
Synonyms:KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:PROTEIN
Mol. Mass.:32031.72
Organism:Homo sapiens (Human)
Description:EBI_12584
Residue:293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARS
DDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGH
YSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPS
AGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDS
CQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
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BDBM33449
n/a
NameBDBM33449
Synonyms:(5-Amino-3-furan-2-yl-[1,2,4]triazol-1-yl)-p-tolyl-methanone | MLS000527907 | SMR000120481 | [5-amino-3-(2-furanyl)-1,2,4-triazol-1-yl]-(4-methylphenyl)methanone | [5-amino-3-(2-furyl)-1,2,4-triazol-1-yl]-(p-tolyl)methanone | [5-amino-3-(furan-2-yl)-1,2,4-triazol-1-yl]-(4-methylphenyl)methanone | [5-azanyl-3-(furan-2-yl)-1,2,4-triazol-1-yl]-(4-methylphenyl)methanone | cid_828590
TypeSmall organic molecule
Emp. Form.C14H12N4O2
Mol. Mass.268.2707
SMILESCc1ccc(cc1)C(=O)n1nc(nc1N)-c1ccco1
Structure
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