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TargetM17 leucyl aminopeptidase
LigandBDBM34324
Substrate/Competitorn/a
Meas. Tech.Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP)
IC50 9620±n/a nM
Citation PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
M17 leucyl aminopeptidase
Name:M17 leucyl aminopeptidase
Synonyms:leucine aminopeptidase
Type:Enzyme Catalytic Domain
Mol. Mass.:67834.32
Organism:Plasmodium falciparum 3D7
Description:gi_124809582
Residue:605
Sequence:
MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
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  Blast E-value cutoff:
BDBM34324
n/a
NameBDBM34324
Synonyms:5-(2,3-dimethylanilino)-3H-1,3,4-thiadiazole-2-thione | 5-[(2,3-dimethylphenyl)amino]-3H-1,3,4-thiadiazole-2-thione | MLS000055478 | SMR000065985 | cid_2374693
TypeSmall organic molecule
Emp. Form.C10H11N3S2
Mol. Mass.237.344
SMILESCc1cccc(Nc2nnc(S)s2)c1C
Structure
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