| Reaction Details |
|---|
 | Report a problem with these data |
| Target | M17 leucyl aminopeptidase |
|---|
| Ligand | BDBM59801 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) |
|---|
| IC50 | 20550±n/a nM |
|---|
| Citation |  PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| M17 leucyl aminopeptidase |
|---|
| Name: | M17 leucyl aminopeptidase |
|---|
| Synonyms: | leucine aminopeptidase |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 67834.32 |
|---|
| Organism: | Plasmodium falciparum 3D7 |
|---|
| Description: | gi_124809582 |
|---|
| Residue: | 605 |
|---|
| Sequence: | MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
|
|
|
|---|
| BDBM59801 |
|---|
| n/a |
|---|
| Name | BDBM59801 |
|---|
| Synonyms: | 4-(5-sulfanyl-4H-1,2,4-triazol-3-yl)phenol | 4-(5-sulfanylidene-1,2,4-triazolidin-3-ylidene)-1-cyclohexa-2,5-dienone | 4-(5-sulfanylidene-1,2,4-triazolidin-3-ylidene)cyclohexa-2,5-dien-1-one | 4-(5-thioxo-1,2,4-triazolidin-3-ylidene)cyclohexa-2,5-dien-1-one | MLS000547905 | SMR000113306 | cid_5387694 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C8H7N3OS |
|---|
| Mol. Mass. | 193.226 |
|---|
| SMILES | Oc1ccc(cc1)-c1n[nH]c(=S)[nH]1 |
|---|
| Structure | 
|
|---|
Search and Browse
