| Reaction Details |
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 | Report a problem with these data |
| Target | M17 leucyl aminopeptidase |
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| Ligand | BDBM51992 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) |
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| IC50 | 13350±n/a nM |
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| Citation |  PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| M17 leucyl aminopeptidase |
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| Name: | M17 leucyl aminopeptidase |
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| Synonyms: | leucine aminopeptidase |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 67834.32 |
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| Organism: | Plasmodium falciparum 3D7 |
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| Description: | gi_124809582 |
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| Residue: | 605 |
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| Sequence: | MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
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| BDBM51992 |
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| n/a |
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| Name | BDBM51992 |
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| Synonyms: | 3-[[(E)-[2-(4-bromobenzyl)oxybenzylidene]amino]thiocarbamoylamino]benzoic acid | 3-[[[2-(4-bromobenzyl)oxybenzylidene]amino]thiocarbamoylamino]benzoic acid | 3-[[[2-[(4-bromophenyl)methoxy]phenyl]methylideneamino]carbamothioylamino]benzoic acid | 3-[[[2-[[2-[(4-bromophenyl)methoxy]phenyl]methylidene]hydrazinyl]-sulfanylidenemethyl]amino]benzoic acid | 3-{[(2-{2-[(4-bromobenzyl)oxy]benzylidene}hydrazino)carbonothioyl]amino}benzoic acid | MLS000681712 | SMR000312756 | cid_16195462 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H18BrN3O3S |
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| Mol. Mass. | 484.366 |
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| SMILES | OC(=O)c1cccc(NC(=S)NN=Cc2ccccc2OCc2ccc(Br)cc2)c1 |w:12.11| |
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| Structure | 
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